Cardarine (GW-501516)

Available in 10mg Tablets (100 Count Bottle)

The Metabolic Endurance Agent | The Non-Hormonal "Exercise Mimetic"

The 4Balance Codex: The Mitochondrial Engine. A potent, selective PPARδ agonist that bypasses androgen pathways to directly modulate cellular metabolism, shifting energy preference toward fatty acid oxidation and aggressively stimulating mitochondrial biogenesis for superior endurance output.

Product Overview

Cardarine (GW-501516) is often grouped with SARMs for research purposes due to similar applications, but its mechanism is fundamentally different. It is not anabolic and does not bind to androgen receptors. It is a selective agonist of the Peroxisome Proliferator-Activated Receptor-delta (PPARδ).

In research models, PPARδ activation acts as a "master switch" for metabolism, simulating the physiological effects of intense endurance exercise even in sedentary states. 4Balance Peptides offers this powerful metabolic agent in precise, laboratory-grade 10mg tablets, ensuring accurate dosage control for sophisticated research protocols compared to liquid alternatives.

Mechanism of Action: The Metabolic Shift

Cardarine’s value in research stems from its ability to fundamentally alter how the body utilizes energy substrates:

1. PPARδ Activation & AMPK Signaling: By binding to the PPARδ nuclear receptor, Cardarine activates the AMP-activated protein kinase (AMPK) pathway. This pathway is normally triggered by energy deficit during exercise. This activation signals skeletal muscle tissue to shift its preferred fuel source from glucose to stored fatty acids.

2. Enhanced Fatty Acid Oxidation (Fat Loss): Research demonstrates that Cardarine upregulates the expression of genes involved in lipid catabolism. By forcing the body to utilize adipose tissue as primary fuel, it drives significant fat loss in animal models without the need for stimulants or induced caloric deficits.

3. Mitochondrial Biogenesis (Endurance): Perhaps its most profound effect in research is the stimulation of mitochondrial biogenesis—the creation of new mitochondria within muscle cells. Combined with the shift of muscle fibers from glycolytic (fast-twitch) to oxidative (slow-twitch), this results in drastic improvements in oxidative capacity and time-to-exhaustion in endurance tests.

4. Muscle Preservation & Lipid Health: Because Cardarine shifts energy usage toward fat stores, it is researched for its "muscle-sparing" properties during caloric restriction, as the body is less likely to catabolize muscle protein for fuel. Furthermore, clinical studies have shown its ability to improve lipid profiles by raising HDL (good) cholesterol and lowering triglycerides.

Primary Research Applications

In the 4Balance Research Array, Cardarine is the premier agent for studies focused on metabolic efficiency and endurance:

• Maximal Endurance Models: Investigating significant increases in aerobic capacity and delay of fatigue onset independent of training status.

• Aggressive Fat Loss & Recomposition: Studying the mechanisms of shifting substrate utilization to adipose tissue while preserving lean muscle mass.

• Metabolic Syndrome & Dyslipidemia: Researching its potential to correct lipid imbalances and improve insulin sensitivity.

• Cardiovascular Research: Investigating PPARδ agonists for their potential anti-inflammatory effects on vascular endothelium.

Technical Specifications

• Compound Name: GW-501516 (Cardarine / Endurobol)

• Format: Oral Tablets

• Concentration: 10mg per Tablet

• Quantity: 100 Tablets

• Purity: ≥99% (HPLC Verified)

• Mechanism: PPARδ Agonist

• Storage: Store at room temperature, away from direct light and moisture.

DISCLAIMER: FOR LABORATORY RESEARCH USE ONLY. This product is a laboratory chemical intended strictly for in-vitro and in-vivo research and development. It is not a drug, dietary supplement, or treatment for any medical condition. NOT for human consumption, veterinary use, or therapeutic application. Bodily introduction of any kind is strictly prohibited by law. Buyer assumes all responsibility for applicable regulations and appropriate use in a research setting.